1L HER2- GC/GEJC trial design

RATIONALE-305: A global, randomized, double-blind, placebo-controlled, phase 3 trial in nearly 1,000 patients with 1L unresectable or metastatic HER2- GC/GEJC1-3

Key eligibility criteria

Key exclusion criteria

R
1:1
(N=997)

TEVIMBRA
200 mg IV Q3W +
investigator-chosen
platinum- and fluoropyrimidine-based chemotherapy
Q3W (n=501)

Placebo IV Q3W +
investigator-chosen
platinum- and fluoropyrimidine-based chemotherapy
Q3W (n=496)

Treatment until disease progression, intolerable toxicity, or withdrawal for other reasons

Key outcomes

Key efficacy outcome:

Additional efficacy outcomes:

Key secondary outcome:

Image description

Key eligibility criteria: Histologically confirmed 1: GC or GEJC and ECOG PS ≤1 within 7 days prior to randomization

Key exclusion criteria: HER2-positive tumors, and previous treatment for unresectable, locally advanced or metastatic GC or GEJC

997 patients randomized 1:1

Dosing: TEVIMBRA 200 mg IV Q3W + investigator-chosen platinum + fluoropyrimidine-containing chemotherapy (n=501). Placebo IV Q3W + investigator-chosen platinum + fluoropyrimidine-containing chemotherapy (n=496). Treatment until disease progression, intolerable toxicity, or withdrawal for other reasons.

Key efficacy outcome: OS in patients with a PD-L1 score ≥1% Additional efficacy outcomes: PFS, ORR, DOR in patients with a PD-L1 score ≥1%

Key secondary outcome: Safety in the all-comer population

Key efficacy analysis in patients with a PD-L1 score ≥1%*: n=885

Safety analysis population: n=992

The patients of RATIONALE-305 were stratified by:

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Leading Expert Discusses RATIONALE-305 Study Design

Dr. Ronan J. Kelly, MD, MBA, reviews RATIONALE-305, a phase 3 trial that evaluated efficacy and safety outcomes with TEVIMBRA + chemotherapy in patients with 1L, unresectable or metastatic, HER2-negative GC or GEJC.

RATIONALE-305 featured a broad range of patients, including those with difficult-to-treat characteristics3

Nearly half of patients exhibited peritoneal metastases

1L GC/GEJC patient characteristics table

PD-L1 scores were measured in RATIONALE-305 using TAP, which demonstrated substantial concordance with CPS, with ~90% agreement3

You may use your preferred PD-L1 testing method to identify patients in clinical practice

Watch the video below to see how PD-L1 scores were tested for clinical trials with TEVIMBRA.

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Leader in Oncology Discusses PD-L1 Testing (TAP vs CPS)

Ronan J. Kelly, MD, MBA, explains TAP, the PD-L1 expression methodology used in the clinical trials of TEVIMBRA.

Frequently Asked Questions

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RATIONALE-305 was a global, randomized, double-blind, placebo-controlled, phase 3 trial in nearly 1,000 patients with 1L, unresectable or metastatic, HER2- GC or GEJC. The key efficacy outcome was overall survival in patients with a PD-L1 score ≥1%.1,3

*PD-L1 scores were measured in RATIONALE-305 using TAP, which demonstrated substantial concordance with CPS, with ~90% agreement. You may use your preferred PD-L1 testing method to identify patients in clinical practice.3
The key efficacy analysis was a retrospective subgroup analysis of RATIONALE-305 in patients with a PD-L1 score ≥1%. PD-L1–negative patients were excluded from this analysis population due to TEVIMBRA + chemotherapy being indicated in patients whose tumors expressed PD-L1 (≥1). Therefore, the efficacy data shared in this presentation do not reflect the all-comer population.3
The race subcategory “Other” included not reported, unknown, and other.3

1L, first line; CPS, combined positive score; DCR, disease control rate; ECOG, Eastern Cooperative Oncology Group; GC, gastric cancer; GEJC, gastroesophageal junction cancer; HER2, human epidermal growth growth factor 2; IV, intravenous; ORR, overall response rate; OS, overall survival; PD-L1, programmed death ligand 1; PFS, progression-free survival; PS, performance status; Q3W, every 3 weeks; R, randomization; TAP, tumor area positivity.

References: 1. TEVIMBRA. Prescribing Information. BeOne Medicines USA, Inc.; 2026. 2. Qiu MZ, Oh DY, Kato K, et al; RATIONALE-305 Investigators. BMJ. 2024;385:e078876. doi:10.1136/bmj-2023-078876 3. Moehler M, Oh DY, Kato K, et al. Adv Ther. 2025;42(5):2248-2268. doi:10.1007/s12325-025-03133-7

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